Publications

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2023
Zahran, S. S., F. A. Ragab, M. G. El-Gazzar, A. M. Soliman, W. R. Mahmoud, and M. M. Ghorab, "Antiproliferative, antiangiogenic and apoptotic effect of new hybrids of quinazoline-4(3H)-ones and sulfachloropyridazine", European Journal of Medicinal Chemistry, vol. 245, pp. 114912-114930 , 2023.
Oudah, K. H., W. R. Mahmoud, F. M. Awadallah, A. T. Tahe, S. E. - S. Abbas, H. A. Allam, and D. Vu, "Design and synthesis of some new benzoylthioureido benzenesulfonamide derivatives and their analogues as carbonic anhydrase inhibitors", Journal of Enzyme Inhibition, vol. 38, pp. 12-23, 2023.
2022
Aziz, N. A. A. M., R. F. George, K. El-Adl, and W. R. Mahmoud, "Design, synthesis, in silico docking, ADMET and anticancer evaluations of thiazolidine-2,4-diones bearing heterocyclic rings as dual VEGFR-2/ EGFRT790M tyrosine kinase inhibitors", RSC Advances, vol. 12, pp. 12913-12931, 2022.
2021
Fouad, M. A., M. Y. Zaki, R. A. Lotfy, and W. R. Mahmoud, "Insight on a new indolinone derivative as an orally bioavailable lead compound against renal cell carcinoma", Bioorganic Chemistry, vol. 112, pp. 104985-104997, 2021.
Hassan, G. S., H. H. Georgey, E. Z. Mohammed, R. F. George, W. R. Mahmoud, and F. A. Omar, "Mechanistic selectivity investigation and 2D-QSAR study of some new antiproliferative pyrazoles and pyrazolopyridines as potential CDK2 inhibitors", European Journal of Medicinal Chemistry, vol. 218, pp. 11389-113410, 2021.
Mohammed, E. Z., W. R. Mahmoud, R. F. George, G. S. Hassan, F. A. Omar, and H. H. Georgey, "Synthesis, in vitro anticancer activity and in silico studies of certain pyrazole-based derivatives as potential inhibitors of cyclin dependent kinases (CDKs)", Bioorganic Chemistry, vol. 116, pp. 105347-105361, 2021.
2019
Georgey, H. H., F. M. Manhi, W. R. Mahmoud, N. A. Mohamed, E. Berrino, and C. T. Supuran, "1,2,4-Trisubstituted imidazolinones with dual carbonic anhydrase and p38 mitogen-activated protein kinase inhibitory activity", Bioorganic Chemistry, vol. 82, pp. 109-116, 2019.
Mahmoud, W. R., Y. M. Nissan, M. M. Elsawah, R. H. Refaey, M. F. Ragab, and K. M. Amin, "Neurobehavioral investigation and acetylcholinesterase inhibitory activity study for some new coumarin derivatives", European Journal of Medicinal Chemistry, vol. 182, pp. 111651-111666, 2019.
Ibrahim, H. S., M. E. Albakri, W. R. Mahmoud, H. A. Allam, A. M. Reda, and H. A. Abdel-Aziz, "Synthesis and biological evaluation of some novel thiobenzimidazole derivatives as anti-renal cancer agents through inhibition of c-MET kinase", Bioorganic Chemistry, vol. 85, pp. 337-348, 2019.
2018
Ibrahim, H. S., H. A. Allam, W. R. Mahmoud, and A. Bonardi, Dual-tail arylsulfone-based benzenesulfonamides differently match the hydrophobic and hydrophilic halves of human carbonic anhydrases active sites: Selective inhibitors for the tumor-associated hCA IX isoform, , 2018.
Awadallah, F. M., S. Bua, W. R. Mahmoud, and H. H. Nada, Inhibition studies on a panel of human carbonic anhydrases with N1-substituted secondary sulfonamides incorporating thiazolinone or imidazolone-indole tails, , 2018.
2015
Abbas, S. E. - S., E. I. Aly, F. M. Awadallah, and W. R. Mahmoud, 4-Substituted-1-phenyl-1H-pyrazolo[3,4-d]pyrimidine Derivatives: Design, Synthesis, Antitumor and EGFR Tyrosine Kinase Inhibitory Activity, , 2015.
2010
Taliawi, G. M. E., E. I. Ali, G. H. Hegazy, and W. Ramadan, Computer Aided Design, Synthesis and Biological Evaluation of Novel Acridine Derivatives a Topoisomerase I Inhibitors, , 2010.
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