Publications

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George, R. F., M. Kandeel, D. Y. El-Ansary, and A. E. M. Kerdawy, "Some 1,3,5-trisubstituted pyrazoline derivatives targeting breast cancer: Design, synthesis, cytotoxic activity, EGFR inhibition and molecular docking", Bioorganic Chemistry, vol. 99, pp. 103780, 2020.
Abbas, S. E. - S., N. M. Abdel-Gawad, R. F. George, M. A. G. Elyazid, M. A. Zaater, and M. K. El-Ashrey, "Some 2-(4-bromophenoxymethyl)-6-iodo-3-substituted quinazolin-4(3H)ones: Synthesis, cytotoxic activity, EGFR inhibition and molecular docking", Journal of Molecular Structure , vol. 1269 , pp. 133851, 2022.
Mahdally, N. H., R. F. George, M. O. N. A. T. KASHEF, M. Al-Ghobashy, F. E. Murad, and A. S. Attia, "Staquorsin: A Novel Staphylococcus aureus Agr-Mediated Quorum Sensing Inhibitor Impairing Virulence in vivo Without Notable Resistance Development", Frontiers in Microbiology, vol. 12, pp. 700494, 2021.
George, R. F., "Stereoselective synthesis and QSAR study of cytotoxic", Eur.J.Med.Chem, vol. 47, pp. 377-386, 2012.
Mabied, A. F., A. S. Girgis, E. - S. M. Shalaby, R. F. George, B. E. - D. M. El-Gendy, and F. N. Baselious, "Stereoselective Synthesis, Structural and Spectroscopic Study of 4,5,11- Triazatricyclo[6.2.1.0*2,6*]Undec-5-ene", J. Heterocyclic Chem., vol. 53, pp. 1074-1080, 2016.
Srour, A. M., S. S. Panda, A. M. M. Salman, M. A. El-Manawaty, R. F. George, E. S. M. Shalaby, A. N. Fitch, N. G. Fawzy, and A. S. Girgis, "Synthesis & molecular modeling studies of bronchodilatory active indole–pyridine conjugates", Future Medicinal Chemistry, vol. 10, issue 15, pp. 1787–1804, 2018.
George, R. F., E. M. Samir, M. N. Abdelhamed, H. A. Abdel-Aziz, and S. E. S. Abbas, "Synthesis and anti-proliferative activity of some new quinoline based 4,5-dihydropyrazoles and their thiazole hybrids as EGFR inhibitors", Bioorganic Chemistry, vol. 83, pp. 186–197, 2019.
Abbas, S. E. S., R. F. George, E. M. Samir, M. M. A. Aref, and H. A. Abdel-Aziz, "Synthesis and anticancer activity of some pyrido[2,3-d]pyrimidine derivatives as apoptosis inducers and cyclin-dependent kinase inhibitors", Future Medicinal Chemistry, vol. 11, issue 18, pp. 2395–2414, 2019.
Abo-Ashour, M. F., W. M. Eldehna, R. F. George, M. M. Abdel-Aziz, M. A. H. M. O. U. D. M. ELAASSER, S. M. Abou-Seri, and N. A. M. Gawad, "Synthesis and biological evaluation of 2-aminothiazole-thiazolidinone conjugates as potential antitubercular agents", Future Medicinal Chemistry, vol. 10, issue 12, pp. 1405–1419, 2018.
George, R. F., M. A. Fouad, and I. E. O. Gomaa, "Synthesis and cytotoxic activities of some pyrazoline derivatives bearing phenyl pyridazine core as new apoptosis inducers", European Journal of Medicinal Chemistry, vol. 112, pp. 48-59, 2016. riham-marwa_paper.pdf
Girgis, A. S., A. F. Mabied, J. Stawinski, L. Hegazy, R. F. George, H. Farag, E. S. M. Shalaby, and A. I. S. Farag, "Synthesis and DFT studies of an antitumor active spiro-oxindole", New Journal of Chemistry, vol. 39, issue 10, pp. 8017-8027, 2015. new_journal_of_chemistry_2015_39_8017_-_8027.pdf
George, R. F., S. S. Panda, E. - S. M. Shalaby, A. M. Srour, A. I. S. Farag, and A. S. Girgis, "Synthesis and molecular modeling studies of indole-based antitumor agents", RSC Advances, vol. 6, pp. 45434-45451, 2016. rsc_adv._2016_6_45434.pdf
Naumov, R. N., S. S. Panda, A. S. Girgis, R. F. George, M. Farhat, and A. R. Katritzky, "Synthesis and QSAR study of novel anti-inflammatory active mesalazine–metronidazole conjugates", Bioorganic & Medicinal Chemistry Letters, vol. 25, issue 11, pp. 2314–2320, 2015. 57_bioorg._med._chem._lett._2015.pdf
George, R. F., M. F. Said, S. Bua, and C. T. Supuran, "Synthesis and selective inhibitory effects of some 2-oxindole benzenesulfonamide conjugates on human carbonic anhydrase isoforms CA I, CA II, CA IX and CAXII", Bioorganic Chemistry, vol. 95, pp. 103514, 2020.
Allam, H. A., A. A. Kamel, M. El-Daly, and R. F. George, "Synthesis and vasodilator activity of some pyridazin-3(2H)-one based compounds", Future Medicinal Chemistry, vol. 12, issue 1, pp. 37–50, 2020.
El-Aleam, R. A. H., R. F. George, G. S. Hassan, and H. M. Abdel-Rahman, "Synthesis of 1,2,4-triazolo[1,5-a]pyrimidine derivatives: Antimicrobial activity, DNA Gyrase inhibition and molecular docking", Bioorganic Chemistry, vol. 94, pp. 103411, 2020.
Panda, S. S., A. S. Girgis, H. H. Honkanadavar, R. F. George, and A. M. Srour, "Synthesis of new ibuprofen hybrid conjugates as potential anti-inflammatory and analgesic agents", Future Medicinal Chemistry, vol. 12, issue 15, pp. 1369–1386, 2020.
Marwa A Ibrahim, R. F. George, S. M. Abou-Seri, and S. M. El-Moghazy, "Synthesis of new phenolic compounds and biological evaluation as antiproliferative agents", Journal of Chemical Research, vol. 44, issue 3-4, pp. 181– 192, 2020.
George, R. F., S. Bua, C. T. Supuran, and F. M. Awadallah, "Synthesis of some N-aroyl-2-oxindole benzenesulfonamide conjugates with carbonic anhydrase inhibitory activity", Bioorganic Chemistry, vol. 96, pp. 103635, 2020.
Hanna, M. M., N. M. Eid, R. F. George, and H. M. Safwat, "Synthesis of some tropane derivatives of anticipated activity on the reuptake of norepinephrine and /or serotonine", Bioorg.Med.Chem, vol. 15, pp. 7765, 2007.
Samir, N., R. F. George, E. Z. Elrazaz, I. M. Ayoub, E. S. M. Shalaby, J. R. Plaisier, N. Demitri, and M. Wink, "Synthesis of some tropane-based compounds targeting colon cancer", Future Medicinal Chemistry, vol. 12, issue 23, pp. 2123-2140, 2020.
Amin, K. M., M. M. Hanna, H. E. Abo-Youssef, and R. F. George, "Synthesis, analgesic and anti-inflammatory activities evaluation of some bi-,tri- and tetracyclic condensed pyrimidines", Eur.J.Med.Chem, vol. 44, pp. 4572, 2009.
George, R. F., N. Samir, I. M. Ayoub, E. S. M. Shalaby, N. Demitri, and M. Wink, "Synthesis, antiproliferative activity and 2D-QSAR study of some 8-alkyl-2,4-bisbenzylidene-3-nortropinones", Future Medicinal Chemistry, vol. 10, issue 24, pp. 2815–2833, 2018.
Amin, K. M., A. M. Taha, R. F. George, N. M. Mohamed, and F. F. Elsenduny, "Synthesis, antitumor activity evaluation, and DNA-binding study of coumarin-based agents", Archiv der Pharmazie, vol. 351, issue 1, pp. 1700199, 2018.
Safinaz E. Abbas, N. A. M. Gawad, R. F. George, and Y. A. Akar, "Synthesis, antitumor and antibacterial activities of some novel tetrahydrobenzo[4,5]thieno[2,3-d]pyrimidine derivatives", European Journalof Medicinal Chemistry, vol. 65, pp. 195-204, 2013. ejmech6165.pdf