Publications

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A
Abbas, S. E. - S., N. M. Abdel-Gawad, R. F. George, M. A. G. Elyazid, M. A. Zaater, and M. K. El-Ashrey, "Some 2-(4-bromophenoxymethyl)-6-iodo-3-substituted quinazolin-4(3H)ones: Synthesis, cytotoxic activity, EGFR inhibition and molecular docking", Journal of Molecular Structure , vol. 1269 , pp. 133851, 2022.
Abbas, S. E. S., R. F. George, E. M. Samir, M. M. A. Aref, and H. A. Abdel-Aziz, "Synthesis and anticancer activity of some pyrido[2,3-d]pyrimidine derivatives as apoptosis inducers and cyclin-dependent kinase inhibitors", Future Medicinal Chemistry, vol. 11, issue 18, pp. 2395–2414, 2019.
Abo-Ashour, M. F., W. M. Eldehna, R. F. George, M. M. Abdel-Aziz, M. A. H. M. O. U. D. M. ELAASSER, N. A. M. Gawad, A. Gupta, S. Bhakta, and S. M. Abou-Seri, "Design, synthesis and whole cell phenotypic evaluation as a novel class of antimicrobial agents. ", European Journal of Medicinal Chemistry, vol. 160, pp. 49-60, 2018.
Abo-Ashour, M. F., W. M. Eldehna, R. F. George, M. M. Abdel-Aziz, M. A. H. M. O. U. D. M. ELAASSER, S. M. Abou-Seri, and N. A. M. Gawad, "Synthesis and biological evaluation of 2-aminothiazole-thiazolidinone conjugates as potential antitubercular agents", Future Medicinal Chemistry, vol. 10, issue 12, pp. 1405–1419, 2018.
Abo-elmagd, N. E., R. F. George, M. A. Ezzat, and R. K. Arafa, "New 1-Phthalazinone scaffold based compounds: Design, synthesis, cytotoxicity and protein kinase inhibition activity.", Mini-Reviews in Medicinal Chemistry, vol. 18, issue 20, pp. 1759-1774, 2018.
Allam, H. A., A. A. Kamel, M. El-Daly, and R. F. George, "Synthesis and vasodilator activity of some pyridazin-3(2H)-one based compounds", Future Medicinal Chemistry, vol. 12, issue 1, pp. 37–50, 2020.
Amin, K. M., G. H. Hegazy, R. F. George, N. R. Ibrahim, and N. M. Mohamed, "Design, synthesis, and pharmacological characterization of some 2‐substituted‐3‐phenyl‐quinazolin‐4(3H)‐one derivatives as phosphodiesterase inhibitors", Archiv der Pharmazie, vol. 354, pp. e2100051, 2021.
Amin, K. M., A. M. Taha, R. F. George, N. M. Mohamed, and F. F. Elsenduny, "Synthesis, antitumor activity evaluation, and DNA-binding study of coumarin-based agents", Archiv der Pharmazie, vol. 351, issue 1, pp. 1700199, 2018.
Amin, K. M., M. M. Hanna, H. E. Abo-Youssef, and R. F. George, "Synthesis, analgesic and anti-inflammatory activities evaluation of some bi-,tri- and tetracyclic condensed pyrimidines", Eur.J.Med.Chem, vol. 44, pp. 4572, 2009.
B
Bokhita, R. M., S. S. Panda, A. S. Girgis, H. H. Honkanadavar, T. S. Ibrahim, R. F. George, M. O. N. A. T. KASHEF, W. A. L. I. D. FAYAD, R. Sakhuja, E. H. Abdel-Aal, et al., "Flouroquinolone-3-carboxamide amino acid conjugates: Synthesis, antibacterial properties and molecular modeling studies", Medicinal Chemistry, vol. 17, pp. 71-84, 2021.
E
Eid, N. M., and R. F. George, "Facile synthesis of some pyrazoline-based compounds with promising anti-inflammatory activity", Future Medicinal Chemistry, vol. 10, issue 2, pp. 183-199, 2018.
El-Aleam, R. A. H., A. M. Sayed, M. N. Taha, R. F. George, H. H. Georgey, and H. M. Abdel-Rahman, "Design and synthesis of novel benzimidazole derivatives as potential Pseudomonas aeruginosa anti-biofilm agents inhibiting LasR: Evidence from comprehensive molecular dynamics simulation and in vitro investigation", European Journal of Medicinal Chemistry, vol. 241, pp. 114629, 2022.
El-Aleam, R. A. H., R. F. George, G. S. Hassan, and H. M. Abdel-Rahman, "Synthesis of 1,2,4-triazolo[1,5-a]pyrimidine derivatives: Antimicrobial activity, DNA Gyrase inhibition and molecular docking", Bioorganic Chemistry, vol. 94, pp. 103411, 2020.
El-Aleam, A. R. H., R. F. George, K. J. Lee, A. B. Keeton, G. A. Piazza, A. A. Kamel, M. E. El-Daly, G. S. Hassan, and H. M. Abdel-Rahman, "Design and synthesis of 1,2,4-triazolo[1,5-a]pyrimidine derivatives as PDE 4B inhibitors endowed with bronchodilator activity", Archiv der Pharmazie, vol. 352, pp. 1900002, 2019.
El-Aleam, R. A. H., R. F. George, H. H. Georgey, and H. M. Abdel-Rahman, "Bacterial virulence factors: a target for heterocyclic compounds to combat bacterial resistance", RSC Advances, vol. 11, pp. 36459–36482, 2021.
El-Moghazy, S. M., R. F. George, E. E. A. Osman, A. A. Elbatrawy, M. Kissova, A. Colombo, E. Crespan, and G. Maga, "Novel pyrazolo[3,4-d]pyrimidines as dual Src-Abl inhibitors active against mutant form of Abl and the leukemia K-562 cell line", European Journal of Medicinal Chemistry, vol. 123, pp. 1-13, 2016. ahmed_published_article.pdf
Elwaie, T. A., S. E. Abbas, E. I. Aly, R. F. George, H. Ali, N. Kraiouchkine, K. S. Abdelwahed, T. E. Fandy, K. E. A. Sayed, Z. A. Y. Elmageed, et al., "HER2 Kinase-Targeted Breast Cancer Therapy: Design, Synthesis, and In Vitro and In Vivo Evaluation of Novel Lapatinib Congeners as Selective and Potent HER2 Inhibitors with Favorable Metabolic Stability", Journal of Medicinal Chemistry, vol. 63, issue 24, pp. 15906−15945, 2020.
Ewida, M. A., H. A. Ewida, M. S. Ahmed, H. A. Allam, R. I. Elbagary, R. F. George, H. H. Georgey, and H. I. El-Subbagh, "3-Methyl-imidazo[2,1-b]thiazole derivatives as a new class of antifolates: Synthesis, in vitro/in vivo bio-evaluation and molecular modeling simulations", Bioorganic Chemistry, vol. 115, pp. 105205, 2021.
Ewida, M. A., H. A. Ewida, M. S. Ahmed, H. A. Allam, R. I. Elbagary, R. F. George, H. H. Georgey, and H. I. El‐Subbagh, "Nanomolar potency of imidazo[2,1‐b]thiazole analogs as indoleamine 2,3‐dioxygenase inhibitors", Archiv der Pharmazie, vol. 354, pp. e2100202, 2021.
F
Farouk, A. K. B. A. W., H. A. Allam, E. Rashwan, R. F. George, and S. E. - S. Abbas, "Design and synthesis of some new 6-bromo-2-(pyridin-3-yl)-4-substituted quinazolines as multi tyrosine kinase inhibitors", Bioorganic Chemistry, vol. 128, pp. 106099, 2022.
G
George, R. F., M. Kandeel, D. Y. El-Ansary, and A. E. M. Kerdawy, "Some 1,3,5-trisubstituted pyrazoline derivatives targeting breast cancer: Design, synthesis, cytotoxic activity, EGFR inhibition and molecular docking", Bioorganic Chemistry, vol. 99, pp. 103780, 2020.
George, R. F., N. S. M. Ismail, J. Stawinski, and A. S. Girgis, "Design, synthesis and QSAR studies of dispiroindole derivatives as new antiproliferative agents", European Journal of Medicinal Chemistry, vol. 68, pp. 339-351, 2013. eur._j._med._chem._68_339-351_2013.pdf
George, R. F., E. M. Samir, M. N. Abdelhamed, H. A. Abdel-Aziz, and S. E. S. Abbas, "Synthesis and anti-proliferative activity of some new quinoline based 4,5-dihydropyrazoles and their thiazole hybrids as EGFR inhibitors", Bioorganic Chemistry, vol. 83, pp. 186–197, 2019.
George, R. F., and D. O. Saleh, "Synthesis, vasorelaxant activity and 2D-QSAR study of some novel pyridazine derivatives", European Journal of Medicinal Chemistry, vol. 108, pp. 663-673, 2016. full_text_published_article.pdf
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