Publications

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2019
El-Aleam, A. R. H., R. F. George, K. J. Lee, A. B. Keeton, G. A. Piazza, A. A. Kamel, M. E. El-Daly, G. S. Hassan, and H. M. Abdel-Rahman, "Design and synthesis of 1,2,4-triazolo[1,5-a]pyrimidine derivatives as PDE 4B inhibitors endowed with bronchodilator activity", Archiv der Pharmazie, vol. 352, pp. 1900002, 2019.
George, R. F., E. M. Samir, M. N. Abdelhamed, H. A. Abdel-Aziz, and S. E. S. Abbas, "Synthesis and anti-proliferative activity of some new quinoline based 4,5-dihydropyrazoles and their thiazole hybrids as EGFR inhibitors", Bioorganic Chemistry, vol. 83, pp. 186–197, 2019.
Abbas, S. E. S., R. F. George, E. M. Samir, M. M. A. Aref, and H. A. Abdel-Aziz, "Synthesis and anticancer activity of some pyrido[2,3-d]pyrimidine derivatives as apoptosis inducers and cyclin-dependent kinase inhibitors", Future Medicinal Chemistry, vol. 11, issue 18, pp. 2395–2414, 2019.
2018
Hassan, G. S., H. H. Georgey, R. F. George, and E. R. Mohammed, "Construction of some cytotoxic agents with aurone and furoaurone scaffolds", Future Medicinal Chemistry, vol. 18, issue 1, pp. 27-52, 2018.
Ghanem, N. M., F. Farouk, R. F. George, S. E. S. Abbas, and O. M. El-Badry, "Design and synthesis of novel imidazo[4,5-b]pyridine based compounds as potent anticancer agents with CDK9 inhibitory activity", Bioorganic Chemistry, vol. 80, pp. 565–576, 2018.
Abo-Ashour, M. F., W. M. Eldehna, R. F. George, M. M. Abdel-Aziz, M. A. H. M. O. U. D. M. ELAASSER, N. A. M. Gawad, A. Gupta, S. Bhakta, and S. M. Abou-Seri, "Design, synthesis and whole cell phenotypic evaluation as a novel class of antimicrobial agents. ", European Journal of Medicinal Chemistry, vol. 160, pp. 49-60, 2018.
George, R. F., "Facile synthesis of simple 2-oxindole-based compounds with promising antiproliferative activity", Future Medicinal Chemistry, vol. 10, issue 3, pp. 269-282, 2018.
Eid, N. M., and R. F. George, "Facile synthesis of some pyrazoline-based compounds with promising anti-inflammatory activity", Future Medicinal Chemistry, vol. 10, issue 2, pp. 183-199, 2018.
Rashad, M. S., H. H. Georgey, R. F. George, and N. M. Abdel-Gawad, "Identification of some benzoxazepines as anticancer agents inducing cancer cell apoptosis", Future Medicinal Chemistry, vol. 10, issue 14, pp. 1649–1664, 2018.
Abo-elmagd, N. E., R. F. George, M. A. Ezzat, and R. K. Arafa, "New 1-Phthalazinone scaffold based compounds: Design, synthesis, cytotoxicity and protein kinase inhibition activity.", Mini-Reviews in Medicinal Chemistry, vol. 18, issue 20, pp. 1759-1774, 2018.
Srour, A. M., S. S. Panda, A. M. M. Salman, M. A. El-Manawaty, R. F. George, E. S. M. Shalaby, A. N. Fitch, N. G. Fawzy, and A. S. Girgis, "Synthesis & molecular modeling studies of bronchodilatory active indole–pyridine conjugates", Future Medicinal Chemistry, vol. 10, issue 15, pp. 1787–1804, 2018.
Abo-Ashour, M. F., W. M. Eldehna, R. F. George, M. M. Abdel-Aziz, M. A. H. M. O. U. D. M. ELAASSER, S. M. Abou-Seri, and N. A. M. Gawad, "Synthesis and biological evaluation of 2-aminothiazole-thiazolidinone conjugates as potential antitubercular agents", Future Medicinal Chemistry, vol. 10, issue 12, pp. 1405–1419, 2018.
George, R. F., N. Samir, I. M. Ayoub, E. S. M. Shalaby, N. Demitri, and M. Wink, "Synthesis, antiproliferative activity and 2D-QSAR study of some 8-alkyl-2,4-bisbenzylidene-3-nortropinones", Future Medicinal Chemistry, vol. 10, issue 24, pp. 2815–2833, 2018.
Amin, K. M., A. M. Taha, R. F. George, N. M. Mohamed, and F. F. Elsenduny, "Synthesis, antitumor activity evaluation, and DNA-binding study of coumarin-based agents", Archiv der Pharmazie, vol. 351, issue 1, pp. 1700199, 2018.
Shalaby, E. S. M., A. M. Srour, S. S. Panda, R. F. George, A. N. Fitch, and A. S. Girgis, "Synthesis, X-ray powder diffraction and DFT-D studies of indole-based compounds", Zeitschrift fur Kristallographie - Crystalline Materials, vol. 233, issue 8, pp. 421-427, 2018.
Hassan, G. S., H. H. Georgey, R. F. George, and E. R. Mohamed, "Aurones and furoaurones: Biological activities and synthesis", Bulletin of Faculty of Pharmacy, Cairo University, vol. 56, pp. 121-127, 2018.
2017
Mohamed, A. R., H. H. Georgey, R. F. George, W. I. El-Eraky, D. O. Saleh, and N. A. M. Gawad, "Identification of some novel xanthinebased derivatives with bronchodilator activity", Future Medicinal Chemistry, vol. 9, issue 15, pp. 1731-1747, 2017.
2016
El-Moghazy, S. M., R. F. George, E. E. A. Osman, A. A. Elbatrawy, M. Kissova, A. Colombo, E. Crespan, and G. Maga, "Novel pyrazolo[3,4-d]pyrimidines as dual Src-Abl inhibitors active against mutant form of Abl and the leukemia K-562 cell line", European Journal of Medicinal Chemistry, vol. 123, pp. 1-13, 2016. ahmed_published_article.pdf
Ismail, N. S. M., R. F. George, R. A. T. Serya, F. N. Baselious, M. El-Manawaty, E. S. M. Shalaby, and A. S. Girgis, "Rational design, synthesis and 2D-QSAR studies of antiproliferative tropane-based compounds", RSC Advances, vol. 6, pp. 101911-101923, 2016. rsc_advances_2016_6_101911_-_101923.pdf
Mabied, A. F., A. S. Girgis, E. - S. M. Shalaby, R. F. George, B. E. - D. M. El-Gendy, and F. N. Baselious, "Stereoselective Synthesis, Structural and Spectroscopic Study of 4,5,11- Triazatricyclo[6.2.1.0*2,6*]Undec-5-ene", J. Heterocyclic Chem., vol. 53, pp. 1074-1080, 2016.
George, R. F., M. A. Fouad, and I. E. O. Gomaa, "Synthesis and cytotoxic activities of some pyrazoline derivatives bearing phenyl pyridazine core as new apoptosis inducers", European Journal of Medicinal Chemistry, vol. 112, pp. 48-59, 2016. riham-marwa_paper.pdf
George, R. F., S. S. Panda, E. - S. M. Shalaby, A. M. Srour, A. I. S. Farag, and A. S. Girgis, "Synthesis and molecular modeling studies of indole-based antitumor agents", RSC Advances, vol. 6, pp. 45434-45451, 2016. rsc_adv._2016_6_45434.pdf
George, R. F., and D. O. Saleh, "Synthesis, vasorelaxant activity and 2D-QSAR study of some novel pyridazine derivatives", European Journal of Medicinal Chemistry, vol. 108, pp. 663-673, 2016. full_text_published_article.pdf
2015
Girgis, A. S., A. F. Mabied, J. Stawinski, L. Hegazy, R. F. George, H. Farag, E. S. M. Shalaby, and A. I. S. Farag, "Synthesis and DFT studies of an antitumor active spiro-oxindole", New Journal of Chemistry, vol. 39, issue 10, pp. 8017-8027, 2015. new_journal_of_chemistry_2015_39_8017_-_8027.pdf
Naumov, R. N., S. S. Panda, A. S. Girgis, R. F. George, M. Farhat, and A. R. Katritzky, "Synthesis and QSAR study of novel anti-inflammatory active mesalazine–metronidazole conjugates", Bioorganic & Medicinal Chemistry Letters, vol. 25, issue 11, pp. 2314–2320, 2015. 57_bioorg._med._chem._lett._2015.pdf