Publications

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2023
Oudah, K. H., W. R. Mahmoud, F. M. Awadallah, A. T. Taher, S. E. - S. Abbas, H. A. Allam, D. Vullo, and C. T. Supuran, "Design and synthesis of some new benzoylthioureido benzene sulfonamide derivatives and their analogues as carbonic anhydrase inhibitors", Journal of Enzyme Inhibition and Medicinal Chemistry , vol. 38, issue 1, pp. 12-23, 2023. paper_15.pdf
2022
Farouk, A. K. B. A. W., H. A. Allam, E. Rashwan, R. F. George, and S. E. - S. Abbas, "Design and synthesis of some new 6-bromo-2-(pyridin-3-yl)-4-substituted quinazolines as multi tyrosine kinase inhibitors", Bioorganic Chemistry , vol. 128, pp. 106099, 2022. paper_13.pdf
Najm, M. A. A., W. R. Mahmoud, A. T. Taher, S. E. - S. Abbas, F. M. Awadallah, H. A. Allam, D. Vullo, and C. T. Supuran, "Design and synthesis of some new benzoylthioureido phenyl derivatives targeting carbonic anhydrase enzymes", Journal of Enzyme Inhibition and Medicinal Chemistry , vol. 37, issue 1, pp. 2702-2709, 2022. paper_14.pdf
Ouf, A. M. A., H. A. Allam, M. Kamel, F. A. Ragab, and S. A. Abdel-Aziz, "Design, synthesis, cytotoxic and enzyme inhibitory activities of 1,3,4-oxadiazole and 1,3,4-thiadiazine hybrids against non-small cell lung cancer ", Results in Chemistry , vol. 4, pp. 100373, 2022.
M.Elimam, D., W. M. Eldehna, R. Salem, A. Bonardi, A. Nocentini, S. T.Al-Rashood, M. M. Elaasser, P. Gratteri, C. T.Supuran, and H.A.Allam, "Natural Inspired Ligustrazine-based SLC-0111 Analogues as Novel Carbonic Anhydrase Inhibitors", european journal of medicinal chemistry, vol. 228, pp. 114008, 2022.
2021
Ewida, M. A., H. A. Ewida, M. S. Ahmed, H. A. Allam, R. I. Elbagary, R. F. George, H. H. Georgey, and H. I. El-Subbagh, "3-Methyl-imidazo[2,1-b]thiazole derivatives as a new class of antifolates: Synthesis, in vitro/in vivo bio-evaluation and molecular modeling simulations", Bioorganic Chemistry , vol. 115, pp. 105205, 2021.
Amin, K. M., A. D. E. Rahman, H. A. Allam, and H. H. El-Zoheiry, "Design and synthesis of novel coumarin derivatives as potential acetylcholinesterase inhibitors for Alzheimer's disease’", Bioorganic Chemistry , vol. 110, pp. 104792, 2021.
Eissa, A. A. M., K. F. M. Aljamal, H. S. Ibrahim, and H. A. Allam, "Design and synthesis of novel pyridopyrimidine derivatives with anchoring non-coplanar aromatic extensions of EGFR inhibitory activity", Bioorganic Chemistry , vol. 115, pp. 105318, 2021.
Ewida, M. A., H. A. Ewida, M. S. Ahmed, H. A. Allam, R. I. Elbagary, R. F. George, H. H. Georgey, and H. I. El‐Subbagh, "Nanomolar potency of imidazo[2,1-b]thiazole analogs as indoleamine 2,3-dioxygenase inhibitors", Archiv der Pharmazie, pp. 2100202, 2021.
2020
Allam, H. A., E. E. Aly, A. K. B. A. W. Farouk, E. A. M. Kerdawy, E. Rashwan, and S. E. S. Abbass, "Design and Synthesis of some new 2,4,6-trisubstituted quinazoline EGFR inhibitors as targeted anticancer agents ", Bioorganic Chemistry , vol. 98, pp. 103726, 2020.
Allam, H. A., A. A. Kamel, M. El-Daly, and R. F. George, "Synthesis and vasodilator activity of some pyridazin-3(2H)-one based compounds", Future Medicinal Chemistry , vol. 12(1), pp. 37-50, 2020.
2019
Ibrahima, H. S., M. E. Albakri, W. R. Mahmoud, H. A. Allam, A. M. Reda, and H. A. Abdel-Aziz, "“Synthesis and biological evaluation of some novel thiobenzimidazole derivatives as anti-renal cancer agents through inhibition of c-MET kinase”", Bioorganic Chemistry , vol. 85, pp. 337-348, 2019.
Allam, H. A., S. H. Fahim, M. F.Abo-Ashour, A. Nocentini, M. E. Elbakry, M. A. Abdel Rahman, W. M. Eldehna, H. S. Ibrahim, and C. T. Supuran, "4- ‘Application of hydrazino and hydrazido linkers to connect benzenesulfonamides with hydrophilic/phobic tails for targeting the middle region of human carbonic anhydrases active site: Selective inhibitors of hCA IX’ ", European Journal of Medicinal Chemistry , vol. 179, pp. 547-556, 2019.
Ragab, F. A. F., S. A. Abdel-Aziz, M. Kamel, A. M. A. Ouf, and H. A. Allam, "Design, synthesis and biological evaluation of some new 1,3,4-thiadiazine-thiourea derivatives as potential antitumor agents against non-small cell lung cancer cells’ ", Bioorganic Chemistry , vol. 93, 2019.
2018
Ibrahima, H. S., H. A. Allam, W. R. Mahmoud, A. Bonardicd, A. Nocentinic, P. Gratteri, E. S. Ibrahim, H. A. Abdel-Aziz, and C. T. Supuran, "Dual-tail arylsulfone-based benzenesulfonamides differently match the hydrophobic and hydrophilic halves of human carbonic anhydrases active sites: Selective inhibitors for the tumor-associated hCA IX isoform", European Journal of Chemistry , vol. 152, pp. 1-9, 2018.
2009
and S. M. El-Moghazy Aly, S.E. Abbas, F. A. E. A. E. H. A., Synthesis of some substituted acridine derivatives of anticipated anticancer activity, , 2009.