Publications

Export 24 results:
Sort by: Author Title Type [ Year (Desc)]
2022
Abdelhaleem, E. F., A. S. M. A. A. E. KASSAB, H. B. El-Nassan, and O. M. Khalil, "Design and Synthesis of Novel Celecoxib Analogues with Potential Cytotoxic and Pro-apoptotic Activity against Breast Cancer Cell Line MCF-7", Medicinal Chemistry, vol. 18, pp. 903-914, 2022. d0008c.pdf
Halim, P. A., H. B. El-Nassan, and Y. S. El-Dash, "Design and Synthesis of Novel Ibuprofen Derivatives as Selective COX-2 Inhibitors and Potential Anti-Inflammatory Agents: Evaluation of PGE2, TNF-α, IL-6 and Histopathological Study", Medicinal Chemistry, vol. 18, pp. 427-443, 2022.
application/pdf iconfinal_manuscript.pdf
2021
El-Nassan, H., "Amberlyst 15®: An Efficient Green Catalyst for the Synthesis of Heterocyclic Compounds", Russian Journal of Organic Chemistry, vol. 57, issue 7, pp. 1109-1134, 2021. el-nassan2021_article_amberlyst15anefficientgreencat.pdf
Kamel, M. M., M. K. Abdel-hameid, H. B. El-Nassan, and E. A. E. - Khouly, "Synthesis and Cytotoxic Activity of Novel Mono- and Bis-Indole Derivatives: Analogues of Marine Alkaloid Nortopsentin", Medicinal Chemistry, vol. 17, issue 7, pp. 779 - 789, 2021.
2020
El‑Meligie, S., N. Khalil, H. B. El-Nassan, and A. Ibraheem, "Efcient synthesis of new 3‑amino‑4‑cyanothiophene derivatives", Chemical Papers, vol. 74, pp. 2491-2500, 2020.
application/pdf iconel-meligie2020_article_efficientsynthesisofnew3-amino.pdf
El‑Meligie, S., N. Khalil, H. B. El-Nassan, and A. Ibraheem, "New synthetic approaches to thieno[3,2‑d]pyrimidine and thieno[3,4‑b]pyridine derivatives", Chemical Papers, vol. 74, pp. 2501-2514, 2020.
application/pdf iconel-meligie2020_article_newsyntheticapproachestothieno.pdf
2019
El-Meligie, S. E. M., N. A. Khalil, H. B. El-Nassan, and A. A. M. Ibraheem, "A Review on the Synthetic Routes to β-Keto Amides", Current Organic Chemistry, vol. 23, issue 19, pp. 2005-2015, 2019.
Kamel, M. M., M. K. Abdel-hameid, H. B. El-Nassan, and E. A. E. - Khouly, "Synthesis and Cytotoxicity Evaluation of Novel Indole Derivatives as Potential Anti-Cancer Agents", medicinal chemistry, vol. 15, issue 8, pp. 873-882, 2019.
2018
El-Nassan, H. B., B. H. Naguib, and E. A. Beshay, "Synthesis of new pyridothienopyrimidinone and pyridothienotriazolopyrimidine derivatives as pim-1 inhibitors", Journal of Enzyme Inhibition and Medicinal Chemistry, vol. 33, issue 1, pp. 58-66, 2018. synthesis_of_new_pyridothienopyrimidinone_and_pyridothienotriazolopyrimidine_derivatives_as_pim_1_inhibitors.pdf
2017
Naguib, B. H., H. B. El-Nassan, and T. M. Abdelghany, "Synthesis of new pyridothienopyrimidinone derivatives as Pim-1 inhibitors", Journal of Enzyme Inhibition and Medicinal Chemistry, vol. 32, issue 1, pp. 457-467, 2017. synthesis_of_new_pyridothienopyrimidinone_derivatives_as_pim_1_inhibitors.pdf
2016
Naguib, B., and H. El-Nassan, "Synthesis of New Thieno[2,3-b]pyridine Derivatives as Pim-1 Inhibitors.", J enzyme inhibition and medicinal chemistry, vol. 31, issue 6, pp. 1718-1725, 2016. synthesis_of_new_thieno_2_3_b_pyridine_derivatives_as_pim_1_inhibitors.pdf
Zaher, A., S. Abuel-Maaty, H. El-Nassan, and S. Amer, "Synthesis, Antitumor Screening and cell cycle analysis of Novel Benzothieno[3,2-b]pyran Derivatives", J enzyme inhibition and medicinal chemistry, vol. 31, issue S4, pp. 145-153, 2016. synthesis_antitumor_screening_and_cell_cycle_analysis_of_novel_benzothieno_3_2_b_pyran_derivatives.pdf
2015
undefined, "Synthesis and antitumor activity of tetrahydrocarbazole hybridized with dithioate derivatives", J Enzyme Inhib Med Chem, vol. 30, issue 2, pp. 308-315, 2015. 147563662e20142e922554.pdf
2014
El-Nassan, H. B., "Recent progress in the identification of BRAF inhibitors as anti-cancer agents", Eur. J. Med. Chem., vol. 72, pp. 170-205, 2014. fkgfahvf.pdf
El-Nassan, H. B., "Synthesis and Structure Activity Relationship Study of N-substituted 3,5-diarylidenepiperidin-4-ones as potential antitumor agents", Anti-Cancer Agents Med. Chem., vol. 14, issue 2, pp. 319-330, 2014. modified_el-nassan-ms.3rd_proof.pdf
2013
El-Nassan, H. B., Advances in the discovery of kinesin spindle protein (Eg5) inhibitors as antitumor agents, : Eur. J. Med. Chem. 62, 614-631 , 2013.
Khalil, N. A., E. M. Ahmed, and H. B. El-Nassan, Synthesis, Characterization and Biological Evaluation of Certain 1,3-Thiazolone Derivatives Bearing Pyrazoline Moiety as Potential Anti-breast Cancer Agents, : Med. Chem. Res. 22,1021-1027, 2013.
2012
Khalil, N. A., E. M. Ahmed, H. B. El-Nassan, and A. A. - A. M. Osama K. Ahmed, Synthesis and Biological Evaluation of Novel Pyrazoline Derivatives as Anti-inflammatory and Antioxidant Agents, : Arch. Pharm. Res. 35, 995-1002 (2012), 2012.
Hameid, M. A. E. K., M. D. Mihovilovic, and H. B. El-Nassan, Synthesis of Novel Pyrazolo[3,4-d]pyrimidine Derivatives as Potential Anti-breast Cancer Agents, : Eur. J. Med. Chem. 57, 323-328 (2012), 2012.
2011
El-Enany, M. M., M. M. Kamel, O. M. Khalil, and H. B. El-Nassan, Synthesis and antitumor activity of novel pyrazolo[1,5-a]pyrimidine derivatives, : Eur. J. Chem. 2, 331-336 (2011), 2011.
El-Nassan, H. B., Synthesis and Antitumor Activity of Novel Pyrido[2,3-d][1,2,4]triazolo[4,3-a]pyrimidin-5-one Derivatives, : Eur. J. Med. Chem. 46, 2031-2036 (2011), 2011.
2010
El-Enany, M. M., S. E. M. El-Meligie, N. A. Abdou, and H. B. El-Nassan, Synthesis and Antimicrobial activity of some 3,5-Diaryl-4,5-dihydropyrazole derivatives, : Orient. J. Chem. 26, 1265-1270 (2010) , 2010.
El-Enany, M. M., M. M. Kamel, O. M. Khalil, and H. B. El-Nassan, Synthesis and antitumor activity of novel 6-aryl and 6-alkylpyrazolo [3,4-d]pyrimidin-4-one derivatives, : Eur. J. Med. Chem. 45, 5286-5291 (2010), 2010.
El-Enany, M. M., S. E. M. El-Meligie, N. A. Abdou, and H. B. El-Nassan, Synthesis of pyrazolo[3,4-b]pyridine and pyrido[2`,3`: 3,4] pyrazolo[1,5-a]pyrimidine derivatives, : J. Chem. Res. 34, 470-474 (2010), 2010.
Tourism