Publications

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2020
Oudaha, K. H., M. A. A. Najma, A. B. Roomi, idy Hussein A.Al-sa, and F. M. Awadallah, "THE RECENT PROGRESS OF SULFONAMIDE IN MEDICINAL CHEMISTRY", Systematic reviews in Pharmacy, vol. 11, issue 12, pp. 1473=1477, 2020.
George, R. F., S. Bua, C. T. Supuran, and F. M. Awadallah, "Synthesis of some N-aroyl-2-oxindole benzenesulfonamide conjugates with carbonic anhydrase inhibitory activity", Bioorganic Chemistry, vol. 96, pp. 103635, 2020.
2019
Elmasry, G. F., E. E. Aly, F. M. Awadallah, and S. M. El-Moghazy, "Design and synthesis of novel PARP-1 inhibitors based on pyridopyridazinone scaffold", Bioorganic chemistry, vol. 87, pp. 655-666, 2019.
2018
Ibrahim, H. A., F. M. Awadallah, H. M. Refaat, and K. M. Amin, "Design, synthesis and molecular modeling study for some new 2-substituted benzimidazoles as dual inhibitors for VEGFR-2 and c-Met", Future medicinal chemistry, vol. 10, pp. 493-509, 2018.
Awadallah, F. M., S. Bua, W. R. Mahmoud, H. H. Nada, A. Nocentini, and C. T. Supuran, "Inhibition studies on a panel of human carbonic anhydrases with N1-substituted secondary sulfonamides incorporating thiazolinone or imidazolone-indole tails", Journal of enzyme inhibition and medicinal chemistry, vol. 33, pp. 629-638, 2018.
Ibrahim, H. A., F. M. Awadallah, H. M. Refaat, and K. M. Amin, "Molecular docking simulation, synthesis and 3D pharmacophore studies of novel 2-substituted-5-nitro-benzimidazole derivatives as anticancer agents targeting VEGFR-2 and c-Met", Biooranic Chemistry, vol. 77, pp. 457-470, 2018.
2017
Samir M. El- Moghazy, Fadi M. Awadallah, Essam Eldin A. Osman, and R. I. Ahmed., "Design, synthesis and molecular docking of novel diarylcyclohexenone and diarylindazole derivatives as tubulin polymerization inhibitors", Journal of enzyme inhibition and medicinal chemistry, vol. 32, pp. 176-188, 2017.
2016
Kamilia M. Amin, Flora F. Barsoum, Fadi M. Awadallah, and N. E. Mohamed, "Identification of new potent phthalazine derivatives with VEGFR-2 and EGFR kinase inhibitory activity", European Journal of Medicinal Chemistry, vol. 123, pp. 191-201, 2016. nehal_paper.pdf
2015
Abbas, S. E. - S., E. I. Aly, F. M. Awadallah, and W. R. Mahmoud, "4-Substituted-1-phenyl-1H-pyrazolo[3,4-d]pyrimidine Derivatives: Design, Synthesis, Antitumor and EGFR Tyrosine Kinase Inhibitory Activity", Chemical Biology and Drug Design, pp. 1-15, 2015. EGFR_paper.pdf
Awadallah, F. M., S. M. Abou-Seri, M. M. Abdulla, and H. H. Georgey, "Design and synthesis of potent 1,2,4-trisubstituted imidazolinone derivatives with dual p38aMAPK and ERK1/2 inhibitory activity", European journal of medicinal chemistry, vol. 94, pp. 397-404, 2015. MAPK/ERK.pdf
Amin, K. M., S. M. Abou-Seri, F. M. Awadallah, and M. A. M. Amal A Eissa, Ghaneya S Hassan, "Synthesis and anticancer activity of some 8-substituted-7-methoxy- 2H-chromen-2-one derivatives toward hepatocellular carcinoma HepG2 cells", European Journal of Medicinal Chemistry, vol. 90, pp. 221-231, 2015. Hepatocellular carcinoma.pdf
Awadallah, F. M., T. A. El-Waei, M. M. Hanna, S. E. Abbas, M. Ceruso, B. E. Oz, O. O. Guler, and C. T. Supuran, "Synthesis, carbonic anhydrase inhibition and cytotoxic activity of novel chromone-based sulfonamide derivatives", European Journal of Medicinal Chemistry, vol. 96, pp. 425-435, 2015. Carbonic anhydrase_paper.pdf
Hassan, G. S., F. M. Awdallah, M. T. El-Saadi, A. O. Elgendi, and L. R. Hemeda, "Synthesis of some benzothiazole derivatives evaluated as antimicrobials and antibiofilms", Journal of Chemical and Pharmaceutical Research, vol. 7, pp. 1125-1143, 2015.
2013
Abbas, S. E. - S., F. M. Awadallah, N. A. Ibrahim, and E. G. Said, "Design and Synthesis of Some 3-Substituted-2-[(2,4-dichlorophenoxy)-methyl]quinazolin-4(3H)-one Derivatives as Potential Anticonvulsant Agents", Chem. Pharm. Bull, vol. 61, issue 7, pp. 679–687, 2013.
Kamilia M. Amin, A. A. M. Eissa, S. M. Abou-Seri, and F. M. Awadallah, "Synthesis and biological evaluation of novel coumarin-pyrazoline hybrids endowed with phenylsulfonyl moiety as antitumor agents", Eur. J. Med. Chem, vol. 60, pp. 187-198, 2013.
Awadallah, F. M., Gary A. Piazza, Bernard D. Gary, and J. C. C. Adam B. Keeton, "Synthesis of some dihydropyrimidine-based compounds bearing pyrazoline moiety and evaluation of their antiproliferative activity", Eur. J. Med. Chem., vol. 70, pp. 273-279, 2013.
2012
Safinaz E. Abbas, F. M. Awadallah, N. A. Ibrahim, and E. G. Said, "New quinazolinone-pyrimidine hybrids: Synthesis, anti-inflammatory and ulcerogenicity studies.", Eur. J. Med. Chem, vol. 53, pp. 141-149, 2012.
Nehad A. El-Sayed, F. M. Awadallah, N. A. Ibrahim, and M. T. El-Saadi, "Potential anti-inflammatory activity and ulcerogenicity study of some novel pyrimido[4',5':4,5]pyrimido[1,6-a]azepine derivatives", Med. Chem. Res., vol. 21, pp. 395–405, 2012.
Fadi M. Awadallah, W. I. El-Eraky, and D. O. Saleh, "Synthesis, vasorelaxant activity, and molecular modeling study of some new phthalazine derivatives", Eur. J. Med. Chem, vol. 52, pp. 14-21, 2012.
2011
Safinaz E. Abbas, F. M. Awadallah, N. A. Ibrahim, and Ahmed M. Gouda, "Design, synthesis and preliminary evaluation of some novel [1,4]diazepino [5,6-b]pyrrolizine and 6-(2-oxopyrrolidino)-1H-pyrrolizine derivatives as anticonvulsant agents", Med. Chem. Res, vol. 20, pp. 1015–1023, 2011.
Kamilia M. Amin, F. M. Awadallah, A. A. M. Eissa, and S. M. Abou-Seri, "Design, synthesis and vasorelaxant evaluation of novel coumarin–pyrimidine hybrids.", Bioorg. Med. Chem, vol. 19, pp. 6087-6097, 2011.
Kamilia M. Amin, G. H. Hanan, and F. M. Awadallah, "EGRF tyrosine kinase targeted compounds: Synthesis, Docking study and In-vitro antitumor activity of some new quinazoline and benzo[d]isothiazole derivatives", Med. Chem. Res, vol. 20, pp. 1042–1053, 2011.
2010
Safinaz E. Abbas, F. M. Awadallah, N. A. Ibrahim, and A. M. Gouda, "Novel substituted and fused pyrrolizine derivatives: synthesis, anti-inflammatory and ulcerogenecity studies", Eur. J. Med. Chem, vol. 45, pp. 482-491, 2010.
Nehad A. El-Sayed, F. M. Awadallah, N. A. Ibrahim, and M. T. El-Saadi, "Synthesis, anti-inflammatory and ulcerogenicity studies of some substituted pyrimido[1,6-a]azepine derivatives", Eur. J. Med. Chem, vol. 45, pp. 3147-3154, 2010.
2008
Awadallah, F. M., "Synthesis, pharmacophore modeling, and biological evaluation of novel 5H-thiazolo[3,2-a]pyrimidin-5-one derivatives as 5-HT2A receptor antagonists", Sci. Pharm., vol. 76, pp. 415-438, 2008.
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