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Curriculum Vittae 

Personal Particulars

Name: Bassem Heshmat Naguib Mina

Date of Birth     : 8 February1972

Place of Birth    : Cairo - Egypt                                            

Nationality                 : Egyptian

Marital status    : Married

Contact             : +2-01224491225

E-Mail: bassem.naguib@pharma.cu.edu.eg

                      Bassem.naguib@bue.edu.eg

Title: Associate Professor – Pharmaceutical Organic Chemistry

Institute: Faculty of Pharmacy, Cairo University, Egypt.

               Faculty of Pharmacy, The British University in Egypt.

 

Education  

  • Philosophy Doctor in Pharmaceutical Science (Organic Chemistry)

          Title of thesis: Synthesis and biological evaluation of benzoxazepines

          University: Cairo University-2008

  • Master degree in Pharmaceutical Science (organic Chemistry)

Title of thesis: Pyridinecarbonitrile derivatives as versatile synthons for some heterocyclic compounds of pharmaceutical interest          University: Cairo University-2002

  • Bachelor degree in Pharmaceutical Science

University: Cairo University-1994

 

Published Papers                      

 

 

1-    “Design, synthesis, and anti-MCF-7 activity of new Thieno[2,3-d]Pyrimidinone derivatives as potential breast cancer treatment.”  Amgad Albohy, Mostafa A. Abdelaziz, Hanan H. Kadry and

Bassem H. Naguib

,

Indian Journal of Heterocyclic Chemistry

. 2024; 34: 1-9. (acceptance letter)

2-    “Novel 3,6-disubstituted pyridazine derivatives targeting JNK1 pathway: Scaffold hopping and hybridization-based design, synthesis, molecular modeling, in vitro and in vivo anticancer evaluation.” Mai M. Shaalan, Essam Eldin A. Osman, Yasmeen M. Attia, Olfat A. Hammam, Riham F. George,

Bassem H. Naguib,

ACS Omega

. 2024; 9: 37310-37329

3-    “Fragment-based design and synthesis of coumarin-based thiazoles as dual c-MET/STAT-3 inhibitors for potential antitumor agents.”

Bassem H. Naguib

, Heba A. Elsebaie, Mohamed S. Nafie, Samy Mohamady, Nader, R. Albujuq, Aya Samir Ayed, Dina Nada, Ahmed F. Khalil, Salma M. Hefny, Haytham O. Tawfik, Moataz A. Shaldam.

Bioorganic Chemistry

. 2024;

151:

107682.

4-    “2-Thioxo-3,4-dihydropyrimidine and thiourea endowed with sulfonamide moieties as dual EGFRT790M and VEGFR-2 inhibitors: Design, synthesis, docking, and anticancer evaluations.

Drug development research

Vol 85, 1-21(2024). Mohamed S. A. El-Gaby, Mohamed A. M. Abdel Reheim, Zuhir S. M. Akrim,

Bassem H. Naguib

, Nashwa M. Saleh, Abu Bakr A. A. M. El-Adasy, Khaled El‐Adl and Samy Mohamady.

5-    “Tailored horseshoe-shaped nicotinonitrile scaffold as dual promising c-Met and Pim-1 inhibitors: Design, synthesis, SAR and in silico study”

Bioorganic Chemistry

Vol 143, 106988 (2024). Samy Mohamady, Ahmed F. Khalil,

Bassem H. Naguib

, Mohamed S. Nafie, Haytham O. Tawfik and Moataz A. Shaldam.

6-    “Design and Novel Synthetic Approach Supported with Molecular Docking and Biological Evidence for Naphthoquinone-Hydrazinotriazolothiadiazine Analogs as Potential Anticancer Inhibiting Topoisomerase-IIB”

Bioorganic Chemistry

Vol 96, 103641 (2020). Samy Mohamady, Mahmoud Salama Ahmed, Abdullah Gibriel, Moataz S. Hendy and

Bassem H. Naguib.

7-    “Structure-based drug design, synthesis, In vitro, and In vivo     biological evaluation of indole-based biomimetic analogs targeting estrogen receptor-α inhibition”

European Journal of Medicinal Chemistry

Vol 166, 281-290 (2019). Moataz S. Hendy, Aya A. AliLubna Ahmed, Reham HossamAlaa Mostafa, Mohamed M. Elmazar,

Bassem H. Naguib

, Yasmeen M. Attia, Mahmoud Salama Ahmed.

8-    “Design, Synthesis, Cytotoxic Activity and Apoptosis-inducing Action of Novel Cinnoline Derivatives as Anticancer Agents.”

Anti-Cancer Agents in Medicinal Chemistry

Vol 18 (8), 1208 - 1217 (2018), Manal M. Kandeel, Aliaa M. Kamal,

Bassem H. Naguib

and Marwa S. A. Hassan

9-    “Synthesis of New Pyridothienopyrimidinone and Pyridothieno -triazolopyrimidine Derivatives as Pim-1 Inhibitors.”

Journal of Enzyme Inhibition and Medicinal Chemistry

Vol 33(1), 58-66 (2018), Hala B. El-Nassan,

Bassem H. Naguib

, Engy A. Beshay

 

10-                    “Synthesis of new pyridothienopyrimidinone derivatives as Pim-1 inhibitors.”

Journal of Enzyme Inhibition and Medicinal Chemistry

Vol 32(1), 457-467 (2017),

Bassem H. Naguib

, Hala B. El-Nassan, Abdelghany, T.M.

11-                    “Synthesis of new thieno[2,3-b]pyridine derivatives as pim-1 inhibitors.”,

Journal of Enzyme Inhibition and Medicinal Chemistry

Vol 31(6), 1718-1725 (2016),

Bassem H. Naguib

, Hala B. El-Nassan.

12-                    “Synthesis and anticonvulsant activity of new phenytoin derivatives.”

European Journal of Medicinal Chemistry

Vol 60, 57-63(2013). Samir Botros Salib, Nadia Abdalla Khalil,

Bassem H. Naguib

, Yara Sayed El-Dash.

13-   “Phenytoin-based Bivalent Ligands: Design, Synthesis and anticonvulsant Activity”.

Archives of Pharmacal Research

Vol 35(12), 2105-2116 (2012). Samir Botros Salib, Nadia Abdalla Khalil,

Bassem Heshmat Naguib

, Yara Sayed El-Dash

14-  “Synthesis and tranquillizing effect of new dibenzoxazepines and pyridobenzoxazepines”,

Egyptian Journal of Chemistry

Vol 54(6), 691-701 (2011), S. Botros,

B. H. Naguib

and A. N. Osman

15-     “Synthesis and tranquillizing effect of new 1,4-benzoxazepines”,  

Egyptian Journal of Chemistry

Vol 54(5), 565-578 (2011), S. Botros,

B. H. Naguib

and A. N. Osman

16-     “Pyridine carbonitrile derivatives as versatile synthons for some heterocyclic compounds of pharmaceutical interest”,

Bulletin of the Faculty of Pharmacy, Cairo University

Vol 41 (3) 2003 p.1-11, M. Mohsen Ismail, R. H. Omar, M.M. Said, A. Ahmady, A. H. Omar,

B. H. Naguib.

 

Conferences Attended

 

1- International Congress on Cell Science and Molecular Biology –       Alexandria: (1-2 August 2022)

Design, Synthesis, and In vitro Anticancer activity of Novel 3,6-  Disubstituted Pyridazine derivatives.

2- 9th International Conference-Faculty of Pharmacy-Cairo University

    Title of research: (April 2018)

     Design, synthesis and insilico-molecular modelling for new 1,3,5-   trisubstitutedpyrazole based analogues.

3- 7th International conference on drug discovery and therapy- Sharjah –      Emirates as speaker (February 2016):

Title of speech:

     “Synthesis of novel [2,3-b] pyridine analogs as Pim-1 inhibitors”

4- 4th International Scientific Conference of Faculty of Pharmacy Cairo

    University (April 2013)

   Title of research:

    “Synthesis and Cytotoxic Activity of New Cinnoline Derivatives”

5- 4th International Scientific Conference of Faculty of Pharmacy Cairo

     University (April 2013) – as organizer.

6- 3rd International Scientific Conference of Faculty of Pharmacy Cairo

    University (April 2012)

    Title of research:

   “Synthesis and anticonvulsant activity of new phenytoin derivatives using

      hybrid approach”

7- 3rd International Scientific Conference of Faculty of Pharmacy Cairo

     University (April 2012) – as organizer.

8- Egyptian Pharmaceutical Society XXXII Conference of Pharmaceutical

     Sciences (December 2011)

     Title of research:

    “Phenytoin-based bivalent ligands: Design, synthesis and anticonvulsant

      activity”

 

Teaching interests and responsibilities

 

Teaching interests:

Lectures and practical courses in Organic Chemistry to students in the undergraduate Pharmacy course (BSc Pharm degree course):

* Stereochemistry – Faculty of Pharmacy, Cairo University (2008, 2009, 2010, 2011, 2012, 2013, 2014, 2015)

* Heterocyclic Chemistry & Stereochemistry, Clinical Pharmacy program

   – Faculty of Pharmacy, Cairo University (Fall 2010)

* Aromatic Organic Chemistry & Spectroscopy – Faculty of Pharmacy,

   Nahda University (spring 2009, summer 2011) as part timer

* Heterocyclic Chemistry & Stereochemistry – Faculty of Pharmacy, Nahda

   University (Fall 2010) as part timer

* Aliphatic Organic Chemistry – Faculty of Pharmacy, Nahda University

   (spring 2011) as part timer

* Aliphatic Organic Chemistry – Faculty of Pharmacy, Misr International   University (fall 2011) as part timer

* Aromatic Organic Chemistry & Heterocyclic Chemistry – Faculty of Pharmacy, Misr International University (summer 2011, fall 2011, spring 2012, summer 2012) as part timer

* Aliphatic Organic Chemistry– Faculty of Pharmacy, Future University (fall 2014) as part timer

* Aliphatic, Aromatic Organic Chemistry, Stereochemistry & Heterocyclic Chemistry – Faculty of Pharmacy, The British University in Egypt (fall 2012, spring 2013, up till now)-

 

Applying Interactive learning (online web learning) for the Courses through Cengage Publisher (2018) and McGrew Hill Publisher (2019, 2020)

 

Other responsibilities:

  • Faculty Exam Office – Faculty of Pharmacy, The British University in Egypt, September 2023 – current.
  • Head of “Teaching, learning and assessment strategy” in “self-evaluation committee” belonging to quality assurance unit September 2023-current.
  • Director of Quality Assurance Unit – Faculty of Pharmacy, The British University in Egypt, May 2021 – August 2023.
  • Member in “research ethical committee” from November 2019 - current
  • Coordinator for Purchasing sector, Faculty of Pharmacy– The British University in Egypt, from September 2015 – May 2021.
  • Elected member of The British University of Egypt Senate from 2017 – 2018.
  • Head of “Financial and material resources” in “self-evaluation committee” belonging to quality assurance unit.
  • Head of “questionnaire committee” belonging to quality assurance unit.
  • Member in “internal audit committee” belonging to quality assurance unit.
  • Vice Manager of Microanalytical center, Faculty of Pharmacy– Cairo University, from June 2014 – August 2015
  • Supervisor of NMR spectrometer and IR spectrometer.
  • Assistant vice dean of education and student affairs, Faculty of Pharmacy– Cairo University, from September 2013 – August 2015
  • Assistant vi
    ce dean of graduate and research affairs

    , Faculty of Pharmacy– Cairo University, from September 2011 – August 2013

-        Supervisor of Kialli research laboratory

-        Coordinator in writing research strategic plan for pharmaceutical organic Chemistry department

  • Assistant vice dean of community services

    , Faculty of Pharmacy– Cairo University, from September 2009 – August 2011

-        Member in the committee for preparing Faculty of Pharmacy – Cairo University for accreditation.

  • Preparing infrastructure booklet

 

Supervisor for six Master degree theses.

 

Training

Interactive electronic courses FLDC-Cairo University 17-18 July 2024
Anti-corruption methods FLDC-Cairo University 22-23 January 2024
Problem solving – based Learning FLDC-Cairo University 17-18 January 2024
Egyptian Knowledge Bank (EKB) and searching for sources FLDC-Cairo University 8-9 January 2024
Essentials of Integrated Education FLDC-Cairo University 27-28 December 2023
Critical thinking FLDC-Cairo University 25-26 December 2023
Fundamentals of digital transformation FLDC-Cairo University 31 December 2023
A Sneak Peek into the Revisions to the CAPE

Outcomes and Entrustable Professional Activities (EPAs)

Accreditation Council for Pharmacy Education, USA 17 January 2023
Program and module specs according to competence-based NARS 2017 The British University in Egypt 22 December 2021
4th Computer assisted Drug Design Workshop Faculty of Pharmacy- Kafrelsheikh University. 6-7 November 2021
Enhance student learning through Kahoot Coursera 30 November 2020
Protocols of external review visit: Applied course for HEI NAQAAE 10-3-2018--13-3-2018
Self-evaluation for H.E. Faculties and institutes NAQAAE 20-11-2017--22-11-2017
University code of ethics FLDC-Cairo University 11-10-2017--12-10-2017

Increasing Student Motivation: a Tool to Overcome Classroom Discipline Problems

The British University in Egypt 13 September 2017

Rethinking the way university students are taught

The British University in Egypt 13 September 2017
Managing research team FLDC-Cairo University 6-7-2017--7-7-2017

Enhancing your lecture for active learning

The British University in Egypt 7 September 2016

Effective presentation skills

The British University in Egypt 7 September 2016

Stress management

The British University in Egypt 7 September 2016

Power point tips to create awesome lectures

The British University in Egypt 7 September 2016
Arabic and English editing in scientific research FLDC-Cairo University 18-5-2016---19-5-2016
International publishing of scientific research FLDC-Cairo University 13-8-2016---14-8-2016
Legal and financial aspects in university environment FLDC-Cairo University 11-5-2016---12-5-2016
Strategic planning FLDC-Cairo University 10-8-2015---11-8-2015
Introduction to Avance NMR spectrometer operation Bruker – Zurich  16-3-2015 ---20-3-2015
Exams & Standards Evaluation Process FLDC-Cairo University 7-6-2010—9-6-2010
Effective Presentation Skills FLDC-Cairo University 7-6-2010—9-6-2010
Use of Technology in Teaching FLDC-Cairo University 31-5-2010—2-6-2010
The Credit Hour Systems FLDC-Cairo University 31-5-2010—2-6-2010
Risk, crisis and emergency plan management CICAP-Faculty of Pharmacy- Cairo university 15-4-2010---15-4-2010
Market orientation in higher education institutions CICAP-Faculty of Pharmacy- Cairo university 6-4-2010---6-4-2010
Computer aided drug design using molecular modelling programs CICAP-Faculty of Pharmacy- Cairo university 1-7-2009---2-7-2009
Research Ethics FLDC-Cairo University 11-8-2008—13-8-2008
Communication Skills FLDC-Cairo University 11-8-2008—13-8-2008

 

Languages

English                  : Spoken / Understanding – fluent.

                                 TOEFL (Local)  Score 570

Arabic

                   

: Native.

 

 

 

*Certificates are available upon request.
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